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ING-132Ingredient Research Profile

Gut Health & Digestive

Zinc Carnosine (PepZin GI)

Also known as: PepZin GI · Polaprezinc · Zinc-L-carnosine

●●○Moderate Evidence

A chelate of zinc and carnosine that adheres to the gastric mucosa, protecting and healing the stomach lining. Approved as a drug in Japan for gastric ulcers.

Effective Dose

75mg (37.5mg zinc + 37.5mg carnosine) twice daily

per clinical evidence

Evidence Level

Moderate

Gut Health & Digestive

Mechanism

Gastric mucosal protection, H. pylori inhibition, mucosal healing

primary action

Best For

Gastric ulcers

NSAID-induced gut damage, H. pylori, Leaky gut

This profile is for informational purposes only and does not constitute medical advice. Consult a qualified healthcare professional before starting any supplementation, especially if you have pre-existing conditions or take medications.

What Is Zinc Carnosine (PepZin GI)?

Zinc carnosine (polaprezinc) is a unique chelate where zinc and L-carnosine form a polymeric structure with exceptional gastric mucosal adherence. It is approved as a prescription drug in Japan for gastric ulcers and H. pylori treatment. Athletic use has grown due to evidence for preventing NSAID-induced gastric damage and reducing exercise-induced gut permeability.

How It Works: The Science

Zinc carnosine adheres to the gastric mucosa (particularly at ulcer sites) and slowly releases zinc and carnosine. Zinc supports mucus secretion and tight junction integrity; carnosine scavenges free radicals and inhibits IL-8 production (reducing inflammatory neutrophil recruitment). It also inhibits H. pylori adhesion to gastric epithelium.

Primary Mechanism

Gastric mucosal protection, H. pylori inhibition, mucosal healing

Evidence-Based Benefits

Heals and prevents gastric and duodenal ulcers

strong

Approved drug in Japan — multiple clinical trials demonstrate ulcer healing

Prevents NSAID-induced gastric damage

moderate

Mahmood et al. (2007) — polaprezinc prevented indomethacin-induced gastric mucosal injury

Reduces exercise-induced gut permeability

moderate

Pugh et al. (2017) — reduced gut permeability markers in endurance athletes

Dosage Guide

Effective Dose

75mg (37.5mg zinc + 37.5mg carnosine) twice daily

75mg zinc carnosine (PepZin GI) twice daily between meals or on an empty stomach. Contains ~37.5mg zinc and ~37.5mg carnosine per 75mg. Monitor total zinc intake.

Safety Profile & Side Effects

Safe at recommended doses. Total zinc from all sources should not exceed 40mg/day (UL). Monitor for copper depletion with long-term use. Approved drug in Japan at these doses.

Who Should (and Shouldn't) Take It

Best for
Gastric ulcersNSAID-induced gut damageH. pyloriLeaky gut
Who it's for

Athletes using NSAIDs for pain management (prevents GI side effects), those with ulcers or H. pylori, and anyone with gut permeability concerns from high-volume training.

Frequently Asked Questions

What is the recommended dose of Zinc Carnosine (PepZin GI)?

75mg zinc carnosine (PepZin GI) twice daily between meals or on an empty stomach. Contains ~37.5mg zinc and ~37.5mg carnosine per 75mg. Monitor total zinc intake.

Is Zinc Carnosine (PepZin GI) safe?

Safe at recommended doses. Total zinc from all sources should not exceed 40mg/day (UL). Monitor for copper depletion with long-term use. Approved drug in Japan at these doses.

How does Zinc Carnosine (PepZin GI) work?

Zinc carnosine adheres to the gastric mucosa (particularly at ulcer sites) and slowly releases zinc and carnosine. Zinc supports mucus secretion and tight junction integrity; carnosine scavenges free radicals and inhibits IL-8 production (reducing inflammatory neutrophil recruitment). It also inhibits H. pylori adhesion to gastric epithelium.

Who should take Zinc Carnosine (PepZin GI)?

Athletes using NSAIDs for pain management (prevents GI side effects), those with ulcers or H. pylori, and anyone with gut permeability concerns from high-volume training.

Related Ingredients

Zinc (Bisglycinate / Picolinate)Probiotics (Lactobacillus / Bifidobacterium)L-GlutamineCollagen Peptides (Type I/III)

Medical Disclaimer

Ingredient profiles are for informational purposes only and do not constitute medical advice. Consult a qualified healthcare professional before starting any supplementation, especially if you have pre-existing conditions or take medications. Full disclaimer →