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ING-091Ingredient Research Profile

Vitamins

Folate (Methylfolate / Vitamin B9)

Also known as: Folic acid · Methyltetrahydrofolate · 5-MTHF · Vitamin B9

●●●Strong Evidence

Critical for DNA synthesis and cell division. Folic acid (synthetic) must be converted to the active form — those with MTHFR gene variants should use methylfolate directly.

Effective Dose

400–800mcg / day

per clinical evidence

Evidence Level

Strong

Vitamins

Mechanism

One-carbon metabolism, DNA synthesis, homocysteine remethylation

primary action

Best For

Pregnancy

Cardiovascular health, MTHFR variants, Cell division

This profile is for informational purposes only and does not constitute medical advice. Consult a qualified healthcare professional before starting any supplementation, especially if you have pre-existing conditions or take medications.

What Is Folate (Methylfolate / Vitamin B9)?

Folate (the natural form) and folic acid (synthetic supplement form) are both forms of vitamin B9. They are essential for one-carbon metabolism — the transfer of single-carbon groups in DNA synthesis, repair, and methylation reactions. Neural tube defects from folate deficiency in early pregnancy are among the most preventable birth defects.

How It Works: The Science

Folate is reduced to tetrahydrofolate (THF) and carries one-carbon units for purine and thymidylate synthesis (DNA building blocks) and for remethylation of homocysteine to methionine (with B12). The MTHFR C677T polymorphism (present in ~10–15% of people) impairs folic acid conversion — methylfolate (5-MTHF) bypasses this step.

Primary Mechanism

One-carbon metabolism, DNA synthesis, homocysteine remethylation

Evidence-Based Benefits

Prevents neural tube defects in early pregnancy

strong

400–800mcg/day periconceptionally reduces NTD risk by 50–70% — public health consensus

Lowers homocysteine (cardiovascular risk marker)

strong

B9 + B12 + B6 combination reduces homocysteine 25–30%

Supports red blood cell maturation

strong

Deficiency causes megaloblastic anaemia — corrected by supplementation

Dosage Guide

Effective Dose

400–800mcg / day

400mcg/day for general population. 800mcg/day for those trying to conceive. Use 5-MTHF (methylfolate) if you have the MTHFR C677T or A1298C variant — folic acid may partially accumulate unmetabolised in these individuals.

Safety Profile & Side Effects

Very safe. Folic acid supplementation can mask B12 deficiency — always pair with B12. Tolerable upper limit: 1000mcg/day (folic acid). No upper limit established for methylfolate.

Who Should (and Shouldn't) Take It

Best for
PregnancyCardiovascular healthMTHFR variantsCell division
Who it's for

All women of reproductive age (mandatory peri-conception), those with MTHFR variants, anyone with elevated homocysteine, and vegans (low dietary folate from fortified foods may be insufficient).

Frequently Asked Questions

What is the recommended dose of Folate (Methylfolate / Vitamin B9)?

400mcg/day for general population. 800mcg/day for those trying to conceive. Use 5-MTHF (methylfolate) if you have the MTHFR C677T or A1298C variant — folic acid may partially accumulate unmetabolised in these individuals.

Is Folate (Methylfolate / Vitamin B9) safe?

Very safe. Folic acid supplementation can mask B12 deficiency — always pair with B12. Tolerable upper limit: 1000mcg/day (folic acid). No upper limit established for methylfolate.

How does Folate (Methylfolate / Vitamin B9) work?

Folate is reduced to tetrahydrofolate (THF) and carries one-carbon units for purine and thymidylate synthesis (DNA building blocks) and for remethylation of homocysteine to methionine (with B12). The MTHFR C677T polymorphism (present in ~10–15% of people) impairs folic acid conversion — methylfolate (5-MTHF) bypasses this step.

Who should take Folate (Methylfolate / Vitamin B9)?

All women of reproductive age (mandatory peri-conception), those with MTHFR variants, anyone with elevated homocysteine, and vegans (low dietary folate from fortified foods may be insufficient).

Related Ingredients

Vitamin B12 (Methylcobalamin)Vitamin B6 (Pyridoxal-5-Phosphate)N-Acetyl Cysteine (NAC)

Medical Disclaimer

Ingredient profiles are for informational purposes only and do not constitute medical advice. Consult a qualified healthcare professional before starting any supplementation, especially if you have pre-existing conditions or take medications. Full disclaimer →