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ING-165Ingredient Research Profile

Superfoods & Botanicals

Cinnamon Extract (Ceylon / Cassia)

Also known as: Cinnamomum verum · Ceylon cinnamon · Cinnamomum cassia

●●○Moderate Evidence

Cinnamon polyphenols sensitise insulin receptors and inhibit alpha-glucosidase, reducing post-meal blood glucose. Ceylon cinnamon is preferred over cassia (which is high in liver-toxic coumarin).

Effective Dose

1–3g / day

per clinical evidence

Evidence Level

Moderate

Superfoods & Botanicals

Mechanism

Insulin receptor sensitisation, alpha-glucosidase inhibition, GLUT4 upregulation

primary action

Best For

Blood sugar

Insulin sensitivity, Cholesterol

This profile is for informational purposes only and does not constitute medical advice. Consult a qualified healthcare professional before starting any supplementation, especially if you have pre-existing conditions or take medications.

What Is Cinnamon Extract (Ceylon / Cassia)?

Cinnamon contains procyanidin B-type polymers (A-type polymers in Ceylon cinnamon) that act as insulin sensitisers — activating insulin receptor tyrosine kinase and inhibiting PTPs (protein tyrosine phosphatases that downregulate insulin signalling). Cinnamaldehyde also inhibits alpha-glucosidase, slowing carbohydrate digestion.

How It Works: The Science

Cinnamon polyphenols activate insulin receptor tyrosine kinase, amplifying the insulin signal and increasing GLUT4 translocation to the cell membrane for glucose uptake. They also inhibit alpha-glucosidase and amylase (reducing carbohydrate digestion speed) and reduce gluconeogenesis via hepatic PEPCK inhibition.

Primary Mechanism

Insulin receptor sensitisation, alpha-glucosidase inhibition, GLUT4 upregulation

Evidence-Based Benefits

Reduces fasting blood glucose in T2D and pre-diabetes

moderate

Allen et al. (2013) meta-analysis — significant reduction in fasting glucose at 1–6g/day

Reduces LDL cholesterol and triglycerides

moderate

Khan et al. (2003) — 1–6g/day for 40 days significantly reduced LDL and triglycerides in T2D

Dosage Guide

Effective Dose

1–3g / day

1–3g Ceylon cinnamon powder or extract daily. Cassia cinnamon (Chinese cinnamon, the most common supermarket variety) contains coumarin at potentially liver-toxic levels at these doses — use Ceylon (true cinnamon) for regular supplementation.

Safety Profile & Side Effects

Ceylon cinnamon: safe at recommended doses. Cassia: coumarin content causes hepatotoxicity at doses above 0.1mg/kg/day long-term — limit cassia cinnamon to culinary amounts. May lower blood glucose — monitor in diabetics on medication.

Who Should (and Shouldn't) Take It

Best for
Blood sugarInsulin sensitivityCholesterol
Who it's for

Pre-diabetic and diabetic individuals wanting blood sugar support alongside dietary change. Choose Ceylon cinnamon or water-extracted cassia (low coumarin) for supplementation.

Frequently Asked Questions

What is the recommended dose of Cinnamon Extract (Ceylon / Cassia)?

1–3g Ceylon cinnamon powder or extract daily. Cassia cinnamon (Chinese cinnamon, the most common supermarket variety) contains coumarin at potentially liver-toxic levels at these doses — use Ceylon (true cinnamon) for regular supplementation.

Is Cinnamon Extract (Ceylon / Cassia) safe?

Ceylon cinnamon: safe at recommended doses. Cassia: coumarin content causes hepatotoxicity at doses above 0.1mg/kg/day long-term — limit cassia cinnamon to culinary amounts. May lower blood glucose — monitor in diabetics on medication.

How does Cinnamon Extract (Ceylon / Cassia) work?

Cinnamon polyphenols activate insulin receptor tyrosine kinase, amplifying the insulin signal and increasing GLUT4 translocation to the cell membrane for glucose uptake. They also inhibit alpha-glucosidase and amylase (reducing carbohydrate digestion speed) and reduce gluconeogenesis via hepatic PEPCK inhibition.

Who should take Cinnamon Extract (Ceylon / Cassia)?

Pre-diabetic and diabetic individuals wanting blood sugar support alongside dietary change. Choose Ceylon cinnamon or water-extracted cassia (low coumarin) for supplementation.

Related Ingredients

BerberineChromium (Picolinate)Gymnema SylvestreBitter Melon (Karela)

Medical Disclaimer

Ingredient profiles are for informational purposes only and do not constitute medical advice. Consult a qualified healthcare professional before starting any supplementation, especially if you have pre-existing conditions or take medications. Full disclaimer →